Adverse Drug Reaction Classification System

Pharmaceutical Information
Drug Name Tenecteplase
Drug ID BADD_D02152
Description Tenecteplase is a tissue plasminogen activator (tPA) developed from modifications of natural human tPA complementary DNA (cDNA). It is a 527 amino acid with a substitution of threonine 103 with asparagine and substitution of asparagine 117 with glutamine within the kringle 1 domain, and a tetra-alanine substitution at amino acids 296-299 in the protease domain.
Indications and Usage For treatment of myocardial infarction and lysis of intracoronary emboli
Marketing Status Prescription
ATC Code B01AD11
DrugBank ID DB00031
KEGG ID D06070
MeSH ID D000077785
PubChem ID Not Available
TTD Drug ID D0FX8A
NDC Product Code 50242-120
Synonyms Tenecteplase | Metalyse | TNKase
Chemical Information
Molecular Formula Not Available
CAS Registry Number 191588-94-0
SMILES Not Available
Chemical Structure
ADR Related Proteins Induced by Drug
ADR Term Protein Name UniProt AC TTD Target ID PMID
Not AvailableNot AvailableNot AvailableNot AvailableNot Available
ADRs Induced by Drug
ADR Term ADReCS ID ADR Frequency (FAERS) ADR Severity Grade (FAERS) ADR Severity Grade (CTCAE)
Anaphylactic reaction24.06.03.006; 10.01.07.001--
Angioedema23.04.01.001; 10.01.05.009--Not Available
Arrhythmia02.03.02.001--Not Available
Atrioventricular block02.03.01.002--Not Available
Cardiac arrest02.03.04.001--
Cardiac failure02.05.01.001--
Cardiac tamponade02.06.01.001--
Cardiogenic shock24.06.02.006; 02.05.01.003--Not Available
Cerebrovascular accident24.03.05.001; 17.08.01.007--
Haemorrhage intracranial24.07.04.003; 17.08.01.008--
Hypotension24.06.03.002--
Laryngeal oedema23.04.01.005; 22.04.02.001; 10.01.05.003--
Mitral valve incompetence02.07.01.002--Not Available
Myocardial infarction24.04.04.009; 02.02.02.007--
Myocardial ischaemia02.02.02.008; 24.04.04.010--Not Available
Myocardial rupture12.01.11.002; 02.04.02.002--Not Available
Nausea07.01.07.001--
Pericardial effusion02.06.01.002--
Pericarditis02.06.02.001--
Pulmonary oedema02.05.02.003; 22.01.03.003--
Pyrexia08.05.02.003--
Rash23.03.13.001--Not Available
Thrombosis24.01.01.006--Not Available
Urticaria23.04.02.001; 10.01.06.001--
Vomiting07.01.07.003--
Haemorrhage24.07.01.002--Not Available
Pulseless electrical activity02.03.04.020--Not Available
Embolism24.01.01.009--
Transfusion25.06.01.003--Not Available
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